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João Paulo dos Santos Fernandes

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Universidade Federal de São Paulo (UNIFESP). Campus Diadema. Instituto de Ciências Ambientais, Químicas e Farmacêuticas (ICAQF)  (Institutional affiliation for the last research proposal)
Birthplace: Brazil

João Paulo dos Santos Fernandes holds a BS in Pharmacy from Guarulhos University (2003). He got his MSc degree at the Faculty of Pharmaceutical Sciences, University of São Paulo (2006) in Medicinal Chemistry, working on prodrugs with tuberculostatic activity, and his PhD degree in the same University (FCF / USP - 2012) working on synthesis and development of histaminergic and serotonin receptor ligands. He has worked in several universities in São Paulo, and currently is full-time professor at Federal University of São Paulo (UNIFESP), dedicated to Medicinal Chemistry in the Pharmacy course as well as graduate programs in Pharmaceutical Sciences and Translational Medicine.Develops research projects with design, synthesis and evaluation of novel bioactive compounds in the central nervous system, inflammatory and infectious/neglected diseases. Member of the European Histamine Research Society (EHRS) and Brazilian Association of Pharmaceutical Sciences (ABCF). He is referee of several international journals and member of the editorial board of the journals Pharmaceutics and Journal of Tuberculosis Research. He heads the group of Synthesis of Bioactive Molecules (SiMBio), from the Laboratory of Natural and Synthetic Inputs (LINS) of UNIFESP. (Source: Lattes Curriculum)

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Scientific publications resulting from Research Grants and Scholarships under the grantee's responsibility (23)

(References retrieved automatically from Web of Science and SciELO through information on FAPESP grants and their corresponding numbers as mentioned in the publications by the authors)

Publications23
Citations49
Cit./Article2.1
Data from Web of Science

VARELA, MARINA T.; COSTA-SILVA, THAIS A.; LAGO, JOAO HENRIQUE G.; TEMPONE, ANDRE G.; FERNANDES, JOAO PAULO S.. Evaluation of the antitrypanosoma activity and SAR study of novel LINS03 derivatives. BIOORGANIC CHEMISTRY, v. 89, . Web of Science Citations: 0. (18/03918-2, 16/25028-3, 18/07885-1, 15/23403-9)

CORRE, MICHELLE F.; BALICO-SILVA, ANDRE L.; KISS, DORA J.; FERNANDES, GUSTAVO A. B.; MARASCHIN, JHONATAN C.; PARREIRAS-E-SILVA, LUCAS T.; VARELA, MARINA T.; SIMOES, SARAH C.; BOUVIER, MICHEL; KESERU, GYORGY M.; et al. Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands - Functional characterization and modeling studies on H-3 and H(4 )receptors. Bioorganic & Medicinal Chemistry, v. 30, . Web of Science Citations: 0. (16/24120-3, 17/05441-6, 12/20148-0, 16/25028-3, 18/03918-2, 18/00153-5, 16/08920-0, 16/23139-2)

CORREA, MICHELLE FIDELIS; DOS SANTOS FERNANDES, JOAO PAULO. Targeting the Histamine H-4 Receptor: Future Drugs for Inflammatory Diseases. CURRENT ORGANIC CHEMISTRY, v. 22, n. 17, p. 1663-1672, . Web of Science Citations: 1. (16/25028-3)

VASCONCELOS, CAMILLA I.; VARELA, MARINA T.; TORRECILHAS, ANA C.; FERNANDES, JOAO P. S.. Pyrazinoates as antiparasitic agents against Trypanosoma cruzi. ARCHIV DER PHARMAZIE, v. 351, n. 11, . Web of Science Citations: 0. (16/01917-3, 18/03918-2, 16/25028-3)

SOLIANI, ANDRESSA; KUBOTA, SILVIA MEGUMI; CORREA, MICHELLE FIDELIS; CERUTTI, SUZETE MARIA; FERNANDES, JOAO PAULO S.. Differential contribution of H3R antagonism by LINS01 compounds on memory, anxiety-like behaviour and spontaneous locomotor activity in healthy rats. Behavioural Brain Research, v. 377, . Web of Science Citations: 0. (16/18039-9, 16/25028-3, 16/23139-2)

GINOZA, MILTON; FERNANDES, GUSTAVO A. B.; CORREA, MICHELLE F.; FERNANDES, JOAO PAULO S.. Novel potent vasodilating agents: Evaluation of the activity and potency of LINS01005 and derivatives in rat aorta. European Journal of Pharmaceutical Sciences, v. 143, . Web of Science Citations: 0. (17/05441-6, 16/23139-2, 16/25028-3)

CORREA, MICHELLE FIDELIS; VARELA, MARINA THEMOTEO; BALBINO, ALEKSANDRO MARTINS; TORRECILHAS, ANA CLAUDIA; LANDGRAF, RICHARDT GAMA; PAOLO TRONCONE, LANFRANCO RANIERI; DOS SANTOS FERNANDES, JOAO PAULO. 1-[(2,3-Dihydro-1-benzofuran-2-yl) methyl]piperazines as novel anti-inflammatory compounds: Synthesis and evaluation on H3R/H4R. CHEMICAL BIOLOGY & DRUG DESIGN, v. 90, n. 2, p. 317-322, . (14/16564-3, 13/18897-7, 13/20479-9)

VARELA, MARINA T.; LIMA, MARTA L.; GALUPPO, MARIANA K.; TEMPONE, ANDRE G.; DE OLIVEIRA, ALBERTO; LAGO, JOAO HENRIQUE G.; FERNANDES, JOAO PAULO S.. New alkenyl derivative from Piper malacophyllum and analogues: Antiparasitic activity against Trypanosoma cruzi and Leishmania infantum. CHEMICAL BIOLOGY & DRUG DESIGN, v. 90, n. 5, p. 1007-1011, . (16/00195-4, 12/18756-1, 15/11936-2, 13/50228-8)

CORREA, MICHELLE F.; BARBOSA, ALEFE J. R.; TEIXEIRA, LARISSA B.; DUARTE, DIEGO A.; SIMOES, SARAH C.; PARREIRAS-E-SILVA, LUCAS T.; BALBINO, ALEKSANDRO M.; LANDGRAF, RICHARDT G.; BOUVIER, MICHEL; COSTA-NETO, CLAUDIO M.; et al. Pharmacological Characterization of 5-Substituted 1-[(2,3-dihydro-1-benzofuran-2-yl)methyl]piperazines: Novel Antagonists for the Histamine H-3 and H-4 Receptors with Anti-inflammatory Potential. FRONTIERS IN PHARMACOLOGY, v. 8, . (16/23139-2, 12/20148-0, 16/25028-3, 17/02042-3, 13/20479-9)

SEGRETTI, NATANAEL DANTE; SIMOES, CRISTINA KORTSTEE; CORREA, MICHELLE FIDELIS; ANDRES FELLI, VENI MARIA; MIYATA, MARCELO; CHO, SANG HYUN; FRANZBLAU, SCOTT GARY; DOS SANTOS FERNANDES, JOAO PAULO. Antimycobacterial activity of pyrazinoate prodrugs in replicating and non-replicating Mycobacterium tuberculosis. TUBERCULOSIS, v. 99, p. 11-16, . (13/20479-9)

VARELA, MARINA T.; DIAS, ROBERTO Z.; MARTINS, LIGIA F.; FERREIRA, DAIANE D.; TEMPONE, ANDRE G.; UENO, ANDERSON K.; LAGO, JOAO HENRIQUE G.; FERNANDES, JOAO PAULO S.. Gibbilimbol analogues as antiparasitic agents-Synthesis and biological activity against Trypanosoma cruzi and Leishmania (L.) infantum. Bioorganic & Medicinal Chemistry Letters, v. 26, n. 4, p. 1180-1183, . (14/16564-3, 12/18756-1, 13/20479-9, 15/11936-2)

MORAIS, THIAGO R.; ALVES CONSERVA, GEANNE A.; VARELA, MARINA T.; COSTA-SILVA, THAIS A.; THEVENARD, FERNANDA; PONCI, VITOR; FORTUNA, ANA; FALCAO, AMILCAR C.; TEMPONE, ANDRE G.; FERNANDES, JOAO PAULO S.; et al. Improving the drug-likeness of inspiring natural products - evaluation of the antiparasitic activity against Trypanosoma cruzi through semi-synthetic and simplified analogues of licarin A. SCIENTIFIC REPORTS, v. 10, n. 1, . Web of Science Citations: 2. (18/07885-1, 18/10279-6, 16/20633-6, 16/25028-3)

OLIVEIRA, LIDIANE; FERRARINI, MARCIO; DOS SANTOS, ALEXANDRE PAES; VARELA, MARINA THEMOTEO; SANTOS CORREA, ISABELA TERESA; TEMPONE, ANDRE GUSTAVO; MELHEM, MARCIA S. C.; VALLIM, MARCELO A.; FERNANDES, JOAO PAULO S.; PASCON, RENATA C.. Coumaric acid analogues inhibit growth and melanin biosynthesis in Cryptococcus neoformans and potentialize amphotericin B antifungal activity. European Journal of Pharmaceutical Sciences, v. 153, . Web of Science Citations: 0. (18/10279-6, 18/03918-2, 15/04400-9, 16/25028-3, 16/14542-8)

FRANCHIN, TAISA BUSARANHO; ULIAN SILVA, BRUNA CRISTINA; DEGRANDIS, RONE APARECIDO; CORREA, MICHELLE FIDELIS; SIMOES DE QUEIROZ ARANHA, CECILIA MARIA; FERNANDES, JOAO PAULO S.; CAMPOS, MICHEL LEANDRO; PECCININI, ROSANGELA GONCALVES. Assessment of the Physicochemical Properties and Stability for Pharmacokinetic Prediction of Pyrazinoic Acid Derivatives. CURRENT DRUG METABOLISM, v. 21, n. 9, p. 714-721, . Web of Science Citations: 0. (16/23139-2, 16/25028-3, 16/23229-1)

WALLER, STEFANIE BRESSAN; CLEFF, MARLETE BRUM; RIPOLL, MARCIA KUTSCHER; ARAUJO MEIRELES, MARIO CARLOS; FERRARINI, MARCIO; VARELA, MARINA THEMOTEO; FERNANDES, JOAO PAULO S.. Bioisosteric modification on benzylidene-carbonyl compounds improved the drug-likeness and maintained the antifungal activity against Sporothrix brasiliensis. CHEMICAL BIOLOGY & DRUG DESIGN, . Web of Science Citations: 0. (16/25028-3, 18/03918-2, 19/24028-8)

VARELA, MARINA T.; ROMANELI, MAIARA M.; LIMA, MARTA L.; BORBOREMA, SAMANTA E. T.; TEMPONE, ANDRE G.; FERNANDES, JOAO P. S.. Antiparasitic activity of new gibbilimbol analogues and SAR analysis through efficiency and statistical methods. European Journal of Pharmaceutical Sciences, v. 122, p. 31-41, . Web of Science Citations: 4. (15/23403-9, 16/00195-4, 16/25028-3)

CORREA, MICHELLE FIDELIS; RAMOS BARBOSA, ALEFE JHONATAS; BORGES FERNANDES, GUSTAVO ARIEL; BAKER, JILLIAN G.; DOS SANTOS FERNANDES, JOAO PAULO. Pharmacological and SAR analysis of the LINS01 compounds at the human histamine H-1, H-2, and H-3 receptors. CHEMICAL BIOLOGY & DRUG DESIGN, v. 93, n. 1, p. 89-95, . Web of Science Citations: 2. (16/23139-2, 17/05441-6, 16/25028-3)

VARELA, MARINA THEMOTEO; FERNANDES, JOAO PAULO S.. Natural Products: Key Prototypes to Drug Discovery against Neglected Diseases Caused by Trypanosomatids. Current Medicinal Chemistry, v. 27, n. 13, p. 2133-2146, . Web of Science Citations: 3. (16/00195-4, 16/25028-3)

CORREA, MICHELLE F.; REINER, DAVID; FERNANDES, GUSTAVO A. B.; VARELA, MARINA T.; ARANHA, CECILIA M. S. Q.; STARK, HOLGER; FERNANDES, JOAO PAULO S.. Profiling of LINS01 compounds at human dopamine D-2 and D-3 receptors. JOURNAL OF CHEMICAL SCIENCES, v. 132, n. 1, . Web of Science Citations: 0. (17/05441-6, 18/03918-2, 18/04488-1, 16/25028-3)

LOPES, FLAVIA B.; ARANHA, CECILIA M. S. Q.; FERNANDES, JOAO PAULO S.. Histamine H-3 receptor and cholinesterases as synergistic targets for cognitive decline: Strategies to the rational design of multitarget ligands. CHEMICAL BIOLOGY & DRUG DESIGN, v. 98, n. 2, . Web of Science Citations: 0. (19/23696-7)

CORREA, MICHELLE FIDELIS; RAMOS BARBOSA, ALEFE JHONATAS; SATO, RIE; JUNQUEIRA, LUIS OTAVIO; POLITI, MARIO JOSE; RANDO, DANIELA GONCALES; DOS SANTOS FERNANDES, JOAO PAULO. Factorial design study to access the ``green{''} iodocyclization reaction of 2-allylphenols. GREEN PROCESSING AND SYNTHESIS, v. 5, n. 2, p. 145-151, . Web of Science Citations: 4. (13/01875-0, 13/20479-9)

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