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(Reference retrieved automatically from Web of Science through information on FAPESP grant and its corresponding number as mentioned in the publication by the authors.)

Functionalization of protected tyrosine via Sonogashira reaction: synthesis of 3-(1,2,3-triazolyl)-tyrosine

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Author(s):
Vasconcelos, Stanley N. S. [1] ; Shamim, Anwar [2] ; Ali, Bakhat [1] ; de Oliveira, Isadora M. [3] ; Stefani, Helio A. [1]
Total Authors: 5
Affiliation:
[1] Univ Sao Paulo, Fac Ciencias Farmaceut, Dept Farm, Sao Paulo, SP - Brazil
[2] Univ Sao Paulo, Inst Quim, Sao Paulo, SP - Brazil
[3] Univ Estadual Oeste Parana, Ctr Engn & Ciencias Exatas, Toledo, PR - Brazil
Total Affiliations: 3
Document type: Journal article
Source: MOLECULAR DIVERSITY; v. 20, n. 2, p. 469-481, MAY 2016.
Web of Science Citations: 2
Abstract

1,2,3-Triazol tyrosines were synthesized from tyrosine alkynes that were in turn prepared via Sonogashira cross-coupling reaction. The tyrosine alkynes were subjected to click-chemistry reaction conditions leading to the corresponding 3-(1,2,3-triazolyl)-tyrosines in yields ranging from moderate to good. (AU)

FAPESP's process: 13/17960-7 - Functionalization of 3-iodo-(L)-Tyrosine via Suzuki-Miyaura Reaction Using Potassium Organotrifluoroborate salts
Grantee:Stanley Nunes Siqueira Vasconcelos
Support Opportunities: Scholarships in Brazil - Doctorate
FAPESP's process: 12/00424-2 - Synthesis of small libraries using potassium Organotrifluoroborates in Suzuki-Miyaura reactions
Grantee:Helio Alexandre Stefani
Support Opportunities: Research Projects - Thematic Grants