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(Reference retrieved automatically from Web of Science through information on FAPESP grant and its corresponding number as mentioned in the publication by the authors.)

Synthesis and functionalization of N-sulfinyl imines: Sonogashira reaction and copper-catalyzed azide-alkyne cycloaddition

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Author(s):
Souza, Frederico B. ; Vasconcelos, Stanley N. S. ; Reis, Joel S. ; Pimenta, Daniel C. ; Stefani, Helio
Total Authors: 5
Document type: Journal article
Source: Tetrahedron Letters; v. 58, n. 11, p. 1057-1060, MAR 15 2017.
Web of Science Citations: 1
Abstract

A small library of novel molecules was generated using a rapid and efficient methodology for the synthesis of N-sulfinyl imine triazole compounds. The process involves a coupling step from the Sonogashira cross-coupling reaction and then, in a one-step reaction, deprotection of the trimethylsilyl group and triazole heterocyclic ring formation using a microwave reactor. (C) 2017 Elsevier Ltd. All rights reserved. (AU)

FAPESP's process: 12/00424-2 - Synthesis of small libraries using potassium Organotrifluoroborates in Suzuki-Miyaura reactions
Grantee:Helio Alexandre Stefani
Support Opportunities: Research Projects - Thematic Grants
FAPESP's process: 16/05260-9 - Synthesis and functionalization of vinyl iodide sulfoxides
Grantee:Frederico Bernardes de Souza
Support Opportunities: Scholarships in Brazil - Doctorate (Direct)