Microwave-Assisted Synthesis of β-1,2,3-Triazolyl-α-amino Esters

Amna N. Khan; Stanley N. S. Vasconcelos; Gonzalo Carrau; Hélio A. Stefani

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(Reference retrieved automatically from SciELO through information on FAPESP grant and its corresponding number as mentioned in the publication by the authors.)

Microwave-Assisted Synthesis of β-1,2,3-Triazolyl-α-amino Esters

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Author(s):	Amna N. Khan ^[1] ; Stanley N. S. Vasconcelos ^[2] ; Gonzalo Carrau ^[3] ; Hélio A. Stefani ^[4] Total Authors: 4
Affiliation:	^[1] Universidade de São Paulo. Faculdade de Ciências Farmacêuticas. Departamento de Farmácia - Brasil ^[2] Universidade de São Paulo. Faculdade de Ciências Farmacêuticas. Departamento de Farmácia - Brasil ^[3] Universidade de São Paulo. Faculdade de Ciências Farmacêuticas. Departamento de Farmácia - Brasil ^[4] Universidade de São Paulo. Faculdade de Ciências Farmacêuticas. Departamento de Farmácia - Brasil Total Affiliations: 4
Document type:	Journal article
Source:	Journal of the Brazilian Chemical Society; v. 26, n. 7, p. 1457-1465, 2015-07-00.
Abstract
<p>The reaction of ethyl (<italic>p</italic>-methoxyphenylimino)acetate with propargyl bromide mediated by activated zinc powder afforded alkynyl amine, which was then reacted with a variety of organic azides using a microwave energy source, leading to β-1,2,3-triazolyl-α-amino esters in good yield.</p> (AU)

FAPESP's process:	12/00424-2 - Synthesis of small libraries using potassium Organotrifluoroborates in Suzuki-Miyaura reactions
Grantee:	Helio Alexandre Stefani
Support Opportunities:	Research Projects - Thematic Grants

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